Category: 1753-29-3

Gil, D. L. published the artcileStructure-activity relations of 1,2,3-benzothiadiazoles as synergists for carbaryl against the house fly (Musca domestica), Name: Benzo[d][1,2,3]thiadiazol-5-amine, the publication is Pesticide Biochemistry and Physiology (1976), 6(4), 338-49, database is CAplus.

1,2,3-Benzothiadiazoles (I, R, R1, R2, R3 = H, halogen, NH2, OH, CN, or alkyl) and related compounds were evaluated as carbaryl [63-25-2] synergists against the housefly (M. domestica). Many of these were excellent synergists, the most active being those containing various combinations of halogen, alkyl, or alkoxy substituents in the 5- and/or 6-positions of the ring. Regression anal. on the data from 14 compounds for which substituents constants were available established that synergistic activity can be satisfactorily described by equations in terms of the hydrophobic bonding constant (π) and the homolytic free radical constant (σâ€?. The results with compounds related to the 1,2,3-benzothiadiazoles suggest that synergistic activity is associated primarily with the diazosulfide moiety.

Pesticide Biochemistry and Physiology published new progress about 1753-29-3. 1753-29-3 belongs to thiazole, auxiliary class Other Aromatic Heterocyclic,Amine, name is Benzo[d][1,2,3]thiadiazol-5-amine, and the molecular formula is C6H5N3S, Name: Benzo[d][1,2,3]thiadiazol-5-amine.

Referemce:
https://pubchem.ncbi.nlm.nih.gov/compound/thiazole,
Thiazole | chemical compound | Britannica

Gil, D. L. published the artcileStructure-activity relationships of 1,2,3-benzothiadiazole insecticide synergists as inhibitors of microsomal oxidation, HPLC of Formula: 1753-29-3, the publication is Pesticide Biochemistry and Physiology (1977), 7(2), 183-93, database is CAplus.

The activities of 47 substituted 1,2,3-benzothiadiazoles (I) as inhibitors of microsomal epoxidation and/or hydroxylation in enzyme preparations from rat liver or armyworm (Spodoptera eridania) gut have been evaluated. Many were found to be effective inhibitors of microsomal oxidation, the most active being the 6-butyl [60474-26-2] and 6-propoxy [63226-45-9] derivatives with I50 values of 4.9 × 10-7 and 7.0 × 10-7 M, resp., for the epoxidation reaction. Regression anal. have established that activity of the 5-, 6-, and 5,6-substituted compounds can be satisfactorily described in equations in terms of π2, π, and σ whereas that of the 4-substituted derivatives depends on π and the steric parameter Es.

Pesticide Biochemistry and Physiology published new progress about 1753-29-3. 1753-29-3 belongs to thiazole, auxiliary class Other Aromatic Heterocyclic,Amine, name is Benzo[d][1,2,3]thiadiazol-5-amine, and the molecular formula is C6H5N3S, HPLC of Formula: 1753-29-3.

Referemce:
https://pubchem.ncbi.nlm.nih.gov/compound/thiazole,
Thiazole | chemical compound | Britannica

Chenard, B. L. published the artcileBenzopentathiepins: synthesis via thermolysis of benzothiadiazoles with sulfur, Application of Benzo[d][1,2,3]thiadiazol-5-amine, the publication is Journal of Organic Chemistry (1984), 49(7), 1221-4, database is CAplus.

A general synthesis of benzopentathiepins I (R = H, 6-Cl, 6-CF₃, 5-MeO, 5-Me₂N, 4-Br, 4-CF₃) has been developed by the thermolysis of benzothiadiazoles II with S. Diazabicyclooctane enhances the yield of benzopentathiepin by approx. 2-fold. The scope and limitations of the method are also discussed.

Journal of Organic Chemistry published new progress about 1753-29-3. 1753-29-3 belongs to thiazole, auxiliary class Other Aromatic Heterocyclic,Amine, name is Benzo[d][1,2,3]thiadiazol-5-amine, and the molecular formula is C6H5N3S, Application of Benzo[d][1,2,3]thiadiazol-5-amine.

Referemce:
https://pubchem.ncbi.nlm.nih.gov/compound/thiazole,
Thiazole | chemical compound | Britannica

Chenard, B. L. published the artcileBenzopentathiepins: synthesis via thermolysis of benzothiadiazoles with sulfur, Application of Benzo[d][1,2,3]thiadiazol-5-amine, the publication is Journal of Organic Chemistry (1984), 49(7), 1221-4, database is CAplus.

A general synthesis of benzopentathiepins I (R = H, 6-Cl, 6-CF₃, 5-MeO, 5-Me₂N, 4-Br, 4-CF₃) has been developed by the thermolysis of benzothiadiazoles II with S. Diazabicyclooctane enhances the yield of benzopentathiepin by approx. 2-fold. The scope and limitations of the method are also discussed.

Journal of Organic Chemistry published new progress about 1753-29-3. 1753-29-3 belongs to thiazole, auxiliary class Other Aromatic Heterocyclic,Amine, name is Benzo[d][1,2,3]thiadiazol-5-amine, and the molecular formula is C6H5N3S, Application of Benzo[d][1,2,3]thiadiazol-5-amine.

Referemce:
https://pubchem.ncbi.nlm.nih.gov/compound/thiazole,
Thiazole | chemical compound | Britannica